Choose the experimental features you want to try

This document is an excerpt from the EUR-Lex website

Document 32010R1238

    Regulation (EU) No 1238/2010 of the European Parliament and of the Council of 15 December 2010 amending Annex I to Council Regulation (EEC) No 2658/87 as regards the provision of duty-free treatment for specified pharmaceutical active ingredients bearing an ‘international non-proprietary name’ (INN) from the World Health Organization and specified products used for the manufacture of finished pharmaceuticals

    OJ L 348, 31.12.2010, p. 36–73 (BG, ES, CS, DA, DE, ET, EL, EN, FR, GA, IT, LV, LT, HU, MT, NL, PL, PT, RO, SK, SL, FI, SV)

    Legal status of the document In force

    ELI: http://data.europa.eu/eli/reg/2010/1238/oj

    31.12.2010   

    EN

    Official Journal of the European Union

    L 348/36


    REGULATION (EU) No 1238/2010 OF THE EUROPEAN PARLIAMENT AND OF THE COUNCIL

    of 15 December 2010

    amending Annex I to Council Regulation (EEC) No 2658/87 as regards the provision of duty-free treatment for specified pharmaceutical active ingredients bearing an ‘international non-proprietary name’ (INN) from the World Health Organization and specified products used for the manufacture of finished pharmaceuticals

    THE EUROPEAN PARLIAMENT AND THE COUNCIL OF THE EUROPEAN UNION,

    Having regard to the Treaty on the Functioning of the European Union, and in particular Article 207 thereof,

    Having regard to the proposal from the European Commission,

    After transmission of the draft legislative act to the national parliaments,

    Acting in accordance with the ordinary legislative procedure (1),

    Whereas:

    (1)

    In the course of the Uruguay Round negotiations, the Community and a number of countries agreed that duty-free treatment should be granted to pharmaceutical products falling within the Harmonised System (HS) Chapter 30 and HS headings 2936, 2937, 2939 and 2941 as well as to designated pharmaceutical active ingredients bearing an ‘international non-proprietary name’ (INN) from the World Health Organization, specified salts, esters and hydrates of such INNs, and designated pharmaceutical intermediates used for the production and manufacture of finished pharmaceuticals.

    (2)

    The results of the discussions, as set out in the Record of Discussions, were incorporated into the tariff schedules of the participants annexed to the Marrakesh Protocol to the General Agreement on Tariffs and Trade (GATT) 1994.

    (3)

    Participants concluded that representatives of World Trade Organization (WTO) members, party to the Record of Discussions, would meet under the auspices of the Council for Trade in Goods of the WTO, normally at least once every three years, to review the product coverage with a view to including, by consensus, additional pharmaceutical products for tariff elimination.

    (4)

    Three such reviews have taken place with the result that a certain number of additional INNs and pharmaceutical intermediates used for the production and manufacture of finished pharmaceuticals have been granted duty-free treatment, that some of those intermediates have been transferred to the list of INNs, and that the list of specified prefixes and suffixes for salts, esters or hydrates of INNs has been expanded.

    (5)

    A fourth review was deemed appropriate and was launched in 2009. It concluded that a certain number of additional INNs and pharmaceutical intermediates used for the production and manufacture of finished pharmaceuticals should be granted duty-free treatment, that some of those intermediates already included in the pharmaceutical sectoral arrangement and its revisions should be transferred to the list of INNs, and that the list of specified prefixes and suffixes for salts, esters or hydrates of INNs should be expanded.

    (6)

    Council Regulation (EEC) No 2658/87 of 23 July 1987 on the tariff and statistical nomenclature and on the Common Customs Tariff (2) established the Combined Nomenclature (CN) and set out the conventional duty rates of the Common Customs Tariff.

    (7)

    Regulation (EEC) No 2658/87 should therefore be amended accordingly.

    (8)

    In order to ensure that the measures provided for in this Regulation apply from 1 January 2011, it should enter into force on the day following that of its publication,

    HAVE ADOPTED THIS REGULATION:

    Article 1

    Annexes 3, 4 and 6 of Section II of Part Three of Annex I to Regulation (EEC) No 2658/87 (Lists of pharmaceutical substances which qualify for duty-free treatment) are hereby amended as follows:

    1.

    As from 1 January 2011 the Union shall extend duty-free treatment to the INNs listed in Annex I.

    2.

    As from 1 January 2011 the list of prefixes and suffixes which, in combination with the INNs included in the pharmaceutical sectoral arrangement and its revisions, describe the salts, esters or hydrates of INNs which are also eligible for duty-free treatment, on condition that they are classifiable in the same six-digit HS subheading as the corresponding INN, shall be amended as set out in Annex II.

    3.

    As from 1 January 2011 the Union shall extend duty-free treatment to the pharmaceutical intermediates used in the production and manufacture of finished pharmaceuticals, listed in Annex III.

    4.

    As from 1 January 2011 the pharmaceutical intermediates listed in Annex IV shall be withdrawn from the list of such compounds receiving duty-free treatment.

    Article 2

    This Regulation shall enter into force on the day following that of its publication in the Official Journal of the European Union.

    It shall apply from 1 January 2011.

    This Regulation shall be binding in its entirety and directly applicable in all Member States.

    Done at Strasbourg, 15 December 2010.

    For the European Parliament

    The President

    J. BUZEK

    For the Council

    The President

    O. CHASTEL


    (1)  Position of the European Parliament of 23 November 2010 (not yet published in the Official Journal) and decision of the Council of 10 December 2010.

    (2)   OJ L 256, 7.9.1987, p. 1.


    ANNEX I

    List of international non-proprietary names (INNs) to be added to the list of products receiving duty-free treatment included in Annex 3 to Annex I to Regulation (EEC) No 2658/87

    CN code

    CAS RN

    Name

    2842 90 80

    119175-48-3

    fermagate

    2843 90 90

    759457-82-4

    padeliporfin

    2844 40 30

    123748-56-1

    iodofiltic acid (

    Formula

    )

    2904 10 00

    21668-77-9

    eprodisate

    2906 19 00

    199798-84-0

    elocalcitol

    2909 30 90

    24150-24-1

    terameprocol

    2916 19 95

    81485-25-8

    peretinoin

    2916 39 00

    51543-40-9

    tarenflurbil

    2918 19 98

    174022-42-5

    bevirimat

    2919 90 00

    258516-89-1

    fospropofol

    2920 90 85

    163133-43-5

    naproxcinod

    2921 19 99

    3687-18-1

    tramiprosate

    2922 19 85

    68392-35-8

    afimoxifene

    2922 19 85

    753449-67-1

    ronacaleret

    2922 29 00

    433265-65-7

    faxeladol

    2922 50 00

    121524-08-1

    amibegron

    2922 50 00

    329773-35-5

    cinaciguat

    2922 50 00

    643094-49-9

    fasobegron

    2923 10 00

    856676-23-8

    choline fenofibrate

    2924 29 98

    847353-30-4

    arbaclofen placarbil

    2924 29 98

    194785-19-8

    bedoradrine

    2924 29 98

    194085-75-1

    carisbamate

    2924 29 98

    254750-02-2

    emricasan

    2924 29 98

    355129-15-6

    eprotirome

    2924 29 98

    402567-16-2

    firategrast

    2924 29 98

    478296-72-9

    gabapentin enacarbil

    2924 29 98

    15866-90-7

    incyclinide

    2924 29 98

    202844-10-8

    indantadol

    2924 29 98

    96847-55-1

    levomilnacipran

    2924 29 98

    608137-32-2

    lisdexamfetamine

    2924 29 98

    652990-07-3

    milveterol

    2924 29 98

    181816-48-8

    ombrabulin

    2924 29 98

    289656-45-7

    senicapoc

    2925 19 95

    19171-19-8

    pomalidomide

    2928 00 90

    22033-87-0

    olesoxime

    2928 00 90

    2675-35-6

    sivifene

    2928 00 90

    816458-31-8

    tecovirimat

    2928 00 90

    238750-77-1

    tosedostat

    2928 00 90

    149647-78-9

    vorinostat

    2929 90 00

    31645-39-3

    palifosfamide

    2930 90 99

    608141-41-9

    apremilast

    2930 90 99

    216167-92-9

    camobucol

    2930 90 99

    211513-37-0

    dalcetrapib

    2930 90 99

    69819-86-9

    darinaparsin

    2930 90 99

    488832-69-5

    elesclomol

    2930 90 99

    216167-95-2

    elsibucol

    2930 90 99

    168682-53-9

    ezatiostat

    2930 90 99

    58569-55-4

    metenkefalin

    2930 90 99

    887148-69-8

    monepantel

    2930 90 99

    603139-19-1

    odanacatib

    2930 90 99

    162520-00-5

    salirasib

    2930 90 99

    216167-82-7

    succinobucol

    2930 90 99

    125961-82-2

    tipelukast

    2931 00 99

    125973-56-0

    amsilarotene

    2932 19 00

    253128-41-5

    eribulin

    2932 19 00

    186953-56-0

    pafuramidine

    2932 29 85

    195883-06-8

    omtriptolide

    2932 99 00

    664338-39-0

    arterolane

    2932 99 00

    183133-96-2

    cabazitaxel

    2932 99 00

    401925-43-7

    celivarone

    2932 99 00

    461432-26-8

    dapagliflozin

    2932 99 00

    118457-15-1

    dexnebivolol

    2932 99 00

    156294-36-9

    larotaxel

    2932 99 00

    118457-16-2

    levonebivolol

    2932 99 00

    83461-56-7

    mifamurtide

    2932 99 00

    117570-53-3

    vadimezan

    2933 19 90

    496775-61-2

    eltrombopag

    2933 19 90

    206884-98-2

    niraxostat

    2933 19 90

    410528-02-8

    palovarotene

    2933 19 90

    376592-42-6

    totrombopag

    2933 29 90

    183659-72-5

    catramilast

    2933 29 90

    944263-65-4

    demiditraz

    2933 29 90

    867153-61-5

    dulanermin

    2933 29 90

    320367-13-3

    lixisenatide

    2933 29 90

    698389-00-3

    rolipoltide

    2933 29 90

    697766-75-9

    velafermin

    2933 39 99

    147084-10-4

    alcaftadine

    2933 39 99

    54-96-6

    amifampridine

    2933 39 99

    249921-19-5

    anamorelin

    2933 39 99

    319460-85-0

    axitinib

    2933 39 99

    208110-64-9

    befiradol

    2933 39 99

    330942-05-7

    betrixaban

    2933 39 99

    201034-75-5

    daporinad

    2933 39 99

    209783-80-2

    entinostat

    2933 39 99

    412950-27-7

    goxalapladib

    2933 39 99

    218791-21-0

    imisopasem manganese

    2933 39 99

    103129-82-4

    levamlodipine

    2933 39 99

    154357-42-3

    levonadifloxacin

    2933 39 99

    108147-54-2

    migalastat

    2933 39 99

    453562-69-1

    motesanib

    2933 39 99

    139145-27-0

    parogrelil

    2933 39 99

    459856-18-9

    pexacerfont

    2933 39 99

    706779-91-1

    pimavanserin

    2933 39 99

    362665-56-3

    pitolisant

    2933 39 99

    861151-12-4

    rosonabant

    2933 39 99

    701977-09-5

    taranabant

    2933 39 99

    189950-11-6

    tropantiol

    2933 39 99

    793655-64-8

    vapitadine

    2933 39 99

    139290-65-6

    volinaserin

    2933 49 90

    141388-76-3

    besifloxacin

    2933 49 90

    697761-98-1

    elvitegravir

    2933 49 90

    185055-67-8

    ferroquine

    2933 49 90

    445041-75-8

    intiquinatine

    2933 49 90

    378746-64-6

    nemonoxacin

    2933 49 90

    245765-41-7

    ozenoxacin

    2933 49 90

    412950-08-4

    rilapladib

    2933 49 90

    871224-64-5

    almorexant

    2933 49 90

    863029-99-6

    balamapimod

    2933 49 90

    698387-09-6

    neratinib

    2933 49 90

    154652-83-2

    tezampanel

    2933 49 90

    128253-31-6

    veliflapon

    2933 59 95

    791828-58-5

    aderbasib

    2933 59 95

    840486-93-3

    adipiplon

    2933 59 95

    850649-61-5

    alogliptin

    2933 59 95

    859212-16-1

    bafetinib

    2933 59 95

    380843-75-4

    bosutinib

    2933 59 95

    839712-12-8

    cariprazine

    2933 59 95

    414910-27-3

    casopitant

    2933 59 95

    288383-20-0

    cediranib

    2933 59 95

    849550-05-6

    cevipabulin

    2933 59 95

    827318-97-8

    danusertib

    2933 59 95

    356057-34-6

    darapladib

    2933 59 95

    501000-36-8

    dutacatib

    2933 59 95

    247257-48-3

    fimasartan

    2933 59 95

    3432-99-3

    folitixorin

    2933 59 95

    668270-12-0

    linagliptin

    2933 59 95

    441798-33-0

    macitentan

    2933 59 95

    641571-10-0

    nilotinib

    2933 59 95

    763113-22-0

    olaparib

    2933 59 95

    686344-29-6

    otenabant

    2933 59 95

    625115-55-1

    riociguat

    2933 59 95

    486460-32-6

    sitagliptin

    2933 59 95

    425637-18-9

    sotrastaurin

    2933 59 95

    309913-83-5

    talmapimod

    2933 59 95

    113857-87-7

    talotrexin

    2933 59 95

    274693-27-5

    ticagrelor

    2933 59 95

    306296-47-9

    vicriviroc

    2933 69 80

    775351-65-0

    imeglimin

    2933 79 00

    461443-59-4

    aplaviroc

    2933 79 00

    189691-06-3

    bremelanotide

    2933 79 00

    813452-18-5

    carmegliptin

    2933 79 00

    405169-16-6

    dovitinib

    2933 79 00

    536748-46-6

    eribaxaban

    2933 79 00

    473289-62-2

    ilepatril

    2933 79 00

    180694-97-7

    mimopezil

    2933 79 00

    579475-18-6

    orvepitant

    2933 79 00

    449811-01-2

    pamapimod

    2933 79 00

    248282-01-1

    paquinimod

    2933 79 00

    380917-97-5

    perampanel

    2933 79 00

    552292-08-7

    rolapitant

    2933 79 00

    425386-60-3

    semagacestat

    2933 79 00

    515814-01-4

    voclosporin

    2933 99 80

    481629-87-2

    aleplasinin

    2933 99 80

    394730-60-0

    boceprevir

    2933 99 80

    649735-63-7

    brivanib alaninate

    2933 99 80

    483369-58-0

    denagliptin

    2933 99 80

    284019-34-7

    denibulin

    2933 99 80

    481631-45-2

    diaplasinin

    2933 99 80

    272105-42-7

    disitertide

    2933 99 80

    227318-71-0

    epetirimod

    2933 99 80

    259793-96-9

    favipiravir

    2933 99 80

    871576-03-3

    flovagatran

    2933 99 80

    229305-39-9

    golotimod

    2933 99 80

    258818-34-7

    larazotide

    2933 99 80

    571170-77-9

    laropiprant

    2933 99 80

    616202-92-7

    lorcaserin

    2933 99 80

    868771-57-7

    melogliptin

    2933 99 80

    803712-67-6

    obatoclax

    2933 99 80

    404950-80-7

    panobinostat

    2933 99 80

    625114-41-2

    piragliatin

    2933 99 80

    74847-35-1

    pyronaridine

    2933 99 80

    872178-65-9

    rabeximod

    2933 99 80

    355151-12-1

    rotigaptide

    2933 99 80

    497221-38-2

    rusalatide

    2933 99 80

    187602-11-5

    sofigatran

    2933 99 80

    227318-75-4

    sotirimod

    2933 99 80

    402957-28-2

    telaprevir

    2933 99 80

    848084-83-3

    tigapotide

    2933 99 80

    393105-53-8

    tiplasinin

    2933 99 80

    620948-93-8

    vabicaserin

    2933 99 80

    794466-70-9

    vernakalant

    2934 10 00

    544417-40-5

    capadenoson

    2934 10 00

    302962-49-8

    dasatinib

    2934 10 00

    223132-37-4

    inolitazone

    2934 10 00

    241479-67-4

    isavuconazole

    2934 10 00

    338990-84-4

    isavuconazonium chloride

    2934 10 00

    607723-33-1

    lobeglitazone

    2934 10 00

    280782-97-0

    managlinat dialanetil

    2934 10 00

    790299-79-5

    masitinib

    2934 10 00

    223673-61-8

    mirabegron

    2934 10 00

    501948-05-6

    rosabulin

    2934 10 00

    447406-78-2

    sodelglitazar

    2934 10 00

    760937-92-6

    teneligliptin

    2934 20 80

    848344-36-5

    bentamapimod

    2934 20 80

    870093-23-5

    talarozole

    2934 99 90

    320345-99-1

    aclidinium bromide

    2934 99 90

    222551-17-9

    adoprazine

    2934 99 90

    207623-20-9

    agatolimod

    2934 99 90

    475479-34-6

    aleglitazar

    2934 99 90

    870524-46-2

    amolimogene bepiplasmid

    2934 99 90

    875446-37-0

    anacetrapib

    2934 99 90

    250386-15-3

    apadenoson

    2934 99 90

    541550-19-0

    apilimod

    2934 99 90

    160707-69-7

    apricitabine

    2934 99 90

    147403-03-0

    azilsartan

    2934 99 90

    863031-21-4

    azilsartan medoxomil

    2934 99 90

    757942-43-1

    bederocin

    2934 99 90

    627861-07-8

    beperminogene perplasmid

    2934 99 90

    959961-96-7

    bevasiranib

    2934 99 90

    769901-96-4

    capeserod

    2934 99 90

    868540-17-4

    carfilzomib

    2934 99 90

    872847-66-0

    cenersen

    2934 99 90

    80295-38-1

    conestat alfa

    2934 99 90

    903916-27-8

    custirsen

    2934 99 90

    187865-22-1

    derquantel

    2934 99 90

    134379-77-4

    dexelvucitabine

    2934 99 90

    247046-52-2

    dilopetine

    2934 99 90

    480449-70-5

    edoxaban

    2934 99 90

    188181-42-2

    elacytarabine

    2934 99 90

    98819-76-2

    esreboxetine

    2934 99 90

    763903-67-9

    fosalvudine tidoxil

    2934 99 90

    172673-20-0

    fosaprepitant

    2934 99 90

    522664-63-7

    ibodutant

    2934 99 90

    405159-59-3

    idrabiotaparinux sodium

    2934 99 90

    188116-07-6

    imepitoin

    2934 99 90

    335619-18-6

    inakalant

    2934 99 90

    1391-36-2

    lancovutide

    2934 99 90

    189059-71-0

    lapaquistat

    2934 99 90

    327026-93-7

    lensiprazine

    2934 99 90

    170632-47-0

    lificiguat

    2934 99 90

    852313-25-8

    litenimod

    2934 99 90

    1000120-98-8

    mipomersen

    2934 99 90

    62253-63-8

    nepidermin

    2934 99 90

    26833-87-4

    omacetaxine mepesuccinate

    2934 99 90

    269718-84-5

    pardoprunox

    2934 99 90

    219923-85-0

    pramiconazole

    2934 99 90

    377727-87-2

    preladenant

    2934 99 90

    524684-52-4

    prinaberel

    2934 99 90

    865311-47-3

    quarfloxin

    2934 99 90

    869884-78-6

    radezolid

    2934 99 90

    496054-87-6

    radiprodil

    2934 99 90

    518048-05-0

    raltegravir

    2934 99 90

    787548-03-2

    regrelor

    2934 99 90

    820957-38-8

    retosiban

    2934 99 90

    572924-54-0

    ridaforolimus

    2934 99 90

    128517-07-7

    romidepsin

    2934 99 90

    93265-81-7

    ropidoxuridine

    2934 99 90

    151823-14-2

    sapacitabine

    2934 99 90

    379231-04-6

    saracatinib

    2934 99 90

    791635-59-1

    simotaxel

    2934 99 90

    119567-79-2

    taribavirin

    2934 99 90

    332012-40-5

    telatinib

    2934 99 90

    925681-61-4

    trabedersen

    2934 99 90

    189003-92-7

    trelanserin

    2934 99 90

    296251-72-4

    velimogene aliplasmid

    2934 99 90

    904302-98-3

    viquidacin

    2934 99 90

    872525-61-6

    votucalis

    2934 99 90

    221877-54-9

    zotarolimus

    2935 00 90

    197904-84-0

    apricoxib

    2935 00 90

    769169-27-9

    begacestat

    2935 00 90

    414864-00-9

    belinostat

    2935 00 90

    313682-08-5

    brecanavir

    2935 00 90

    839673-52-8

    cevoglitazar

    2935 00 90

    358970-97-5

    drinabant

    2935 00 90

    865200-20-0

    giripladib

    2935 00 90

    464213-10-3

    ibipinabant

    2935 00 90

    173424-77-6

    laromustine

    2935 00 90

    398507-55-6

    lodenafil carbonate

    2935 00 90

    136564-68-6

    masilukast

    2935 00 90

    170569-88-7

    mavacoxib

    2935 00 90

    862189-95-5

    mirodenafil

    2935 00 90

    439687-69-1

    nelivaptan

    2935 00 90

    691852-58-1

    nesbuvir

    2935 00 90

    778576-62-8

    oglemilast

    2935 00 90

    444731-52-6

    pazopanib

    2935 00 90

    362505-84-8

    relacatib

    2935 00 90

    243984-11-4

    resatorvid

    2935 00 90

    519055-62-0

    tasisulam

    2935 00 90

    186497-07-4

    zibotentan

    2936 29 00

    104121-92-8

    eldecalcitol

    2936 29 00

    31690-09-2

    levomefolic acid

    2937 19 00

    782500-75-8

    albiglutide

    2937 19 00

    348119-84-6

    obinepitide

    2937 19 00

    295350-45-7

    ozarelix

    2937 19 00

    275371-94-3

    taspoglutide

    2937 19 00

    218949-48-5

    tesamorelin

    2937 19 00

    22006-64-0

    tridecactide

    2937 22 00

    132245-57-9

    dexamethasone cipecilate

    2937 22 00

    397864-44-7

    fluticasone furoate

    2937 29 00

    211254-73-8

    lonaprisan

    2937 50 00

    333963-42-1

    cobiprostone

    2937 50 00

    172740-14-6

    posaraprost

    2937 90 00

    834153-87-6

    elagolix

    2937 90 00

    609799-22-6

    tasimelteon

    2937 90 00

    342577-38-2

    velneperit

    2939 19 00

    73232-52-7

    methylnaltrexone bromide

    2939 59 00

    136199-02-5

    rolofylline

    2939 99 00

    850607-58-8

    darotropium bromide

    2939 99 00

    187852-63-7

    delimotecan

    2940 00 00

    9007-72-1

    ferric carboxymaltose

    2940 00 00

    442201-24-3

    remogliflozin etabonate

    2940 00 00

    408504-26-7

    sergliflozin etabonate

    2941 90 00

    467214-20-6

    alvespimycin

    2941 90 00

    677017-23-1

    berubicin

    2941 90 00

    229016-73-3

    ceftaroline fosamil

    2941 90 00

    318498-76-9

    flopristin

    2941 90 00

    145435-72-9

    gamithromycin

    2941 90 00

    325965-23-9

    linopristin

    2941 90 00

    857402-23-4

    retaspimycin

    2941 90 00

    305841-29-6

    sagopilone

    2941 90 00

    75747-14-7

    tanespimycin

    2941 90 00

    328898-40-4

    tildipirosin

    2941 90 00

    222400-20-6

    tomopenem

    2941 90 00

    63409-12-1

    tylvalosin

    3001 90 91

    9041-08-1

    semuloparin sodium

    3002 10 91

    792921-10-9

    abagovomab

    3002 10 91

    910649-32-0

    anrukinzumab

    3002 10 91

    648904-28-3

    bavituximab

    3002 10 91

    402710-27-4

    (light chain)

    402710-25-2

    (heavy chain)

    canakinumab

    3002 10 99

    945228-49-9

    citatuzumab bogatox

    3002 10 91

    880486-59-9

    dacetuzumab

    3002 10 91

    615258-40-7

    denosumab

    3002 10 91

    762260-74-2

    efungumab

    3002 10 91

    89957-37-9

    gantenerumab

    3002 10 91

    680188-33-4

    ibalizumab

    3002 10 91

    477202-00-9

    ipilimumab

    3002 10 91

    640735-09-7

    iratumumab

    3002 10 91

    845816-02-6

    lexatumumab

    3002 10 91

    903512-50-5

    lucatumumab

    3002 10 91

    899796-83-9

    milatuzumab

    3002 10 91

    677010-34-3

    motavizumab

    3002 10 91

    676258-98-3

    naptumomab estafenatox

    3002 10 91

    828933-51-3

    nimotuzumab

    3002 10 91

    949142-50-1

    obinutuzumab

    3002 10 91

    637334-45-3

    ocrelizumab

    3002 10 91

    881191-44-2

    otelixizumab

    3002 10 91

    372075-37-1

    sontuzumab

    3002 10 91

    705287-60-1

    stamulumab

    3002 10 91

    339086-80-5

    tadocizumab

    3002 10 91

    592557-43-2

    (light chain)

    592557-41-0

    (heavy chain)

    tenatumomab

    3002 10 91

    876387-05-2

    teplizumab

    3002 10 91

    918127-53-4

    tigatuzumab

    3002 10 91

    745013-59-6

    tremelimumab

    3002 10 91

    339986-90-2

    tucotuzumab celmoleukin

    3002 10 91

    728917-18-8

    veltuzumab

    3002 10 91

    896731-82-1

    conatumumab

    3002 10 91

    892553-42-3

    etaracizumab

    3002 10 91

    944548-38-3

    foravirumab

    3002 10 91

    944548-37-2

    rafivirumab

    3002 10 91

    880266-57-9

    tanezumab

    3002 10 91

    815610-63-0

    ustekinumab

    3002 10 95

    862111-32-8

    aflibercept

    3002 10 95

    845264-92-8

    atacicept

    3002 10 95

    909110-25-4

    baminercept

    3002 10 95

    9001-27-8

    beroctocog alfa

    3002 10 95

    879555-13-2

    epoetin kappa

    3002 10 95

    762263-14-9

    epoetin theta

    3002 10 95

    501081-76-1

    rilonacept

    3002 10 95

    267639-76-9

    romiplostim

    3002 10 95

    869858-13-9

    thrombin alfa

    3002 10 95

    897936-89-9

    vatreptacog alfa (activated)

    3002 10 95

    472960-22-8

    albinterferon alfa-2b

    3002 10 95

    869881-54-9

    briobacept

    3002 10 95

    606138-08-3

    catridecacog

    3002 10 95

    716840-32-3

    denenicokin

    3002 10 95

    931101-84-7

    troplasminogen alfa

    3002 10 99

    934216-54-3

    alacizumab pegol

    3002 20 00

    181477-43-0

    disomotide

    3002 20 00

    181477-91-8

    ovemotide

    3002 20 00

    915019-08-8

    tertomotide

    3002 20 00

    295371-00-5

    verpasep caltespen

    3002 90 90

    473553-86-5

    alferminogene tadenovec

    3002 90 90

    929881-05-0

    alipogene tiparvovec

    3002 90 90

    600735-73-7

    contusugene ladenovec

    3002 90 90

    851199-59-2

    linaclotide

    3002 90 90

    898830-54-1

    sitimagene ceradenovec

    3002 90 90

    721946-42-5

    transferrin aldifitox

    3507 90 90

    9026-00-0

    bucelipase alfa

    3507 90 90

    885051-90-1

    pegloticase

    3507 90 90

    884604-91-5

    velaglucerase alfa

    3911 90 99

    892497-01-7

    azoximer bromide


    ANNEX II

    List of prefixes and suffixes which, in combination with the INNs of Annex 3 to Annex I to Regulation (EEC) No 2658/87, describe the salts, esters or hydrates of INNs; these salts, esters and hydrates are free of duty, on condition that they are classifiable in the same six-digit HS subheading as the corresponding INN

    The references to ‘International Nonproprietary Names (INN) for pharmaceutical substances, names for radicals and groups, comprehensive list 2004’ are replaced by ‘International Nonproprietary Names (INN) for pharmaceutical substances, names for radicals, groups and others, comprehensive list 2007’.

    The following prefixes or suffixes are added to the list included in Annex 4 to Annex I to Regulation (EEC) No 2658/87:

    Preferred prefix or suffix

    Synonym

    Systematic name when different

    alanetil (INNRG)

     

    [(S)-1-ethoxy-1-oxo-propan-2-yl]amino (INNCN)

    alaninate (INNRG)

     

    L-alaninate (INNCN)

    alapivoxil (INNRG)

     

    L-alanyl, [(2,2-dimethylpropanoyl)oxy]metyl (INNCN)

    aldifitox (INNRG)

     

    (4-iminobutane-1,4-diyl)sulfanediyl[(3RS)-2,5-dioxopyrrolidine-1,3-diyl]-1,3-phenylenecarbonyl and forming an N-benzoyl derivative of a primary amine group of diphtheria [550-L-phenylalanine]toxin from Corynebacterium diphtheriae-(26-560)-peptide (INNCN)

    besudotox (INNRG)

     

    L-lysyl-L-alanyl-L-serylglycylglycine (linker) fusion protein with des-(365-380)-[Asn364,Val407,Ser515,Gln590,Gln606,Arg613]exotoxin A (Pseudomonas aeruginosa)-(251-613)-peptide (toxin with region IA and first 16 residues of region IB deleted) (INNCN)

    ceribate (INNRG)

     

    rac-2,3-dihydroxypropyl carbonate (ester) (INNCN)

    cipecilate (INNRG)

     

    cyclohexanecarboxylate (ester), cyclopropanecarboxylate (ester) (INNCN)

    dalanated (INNRG)

     

    des-B30-alanine (INNCN)

    enacarbil (INNRG)

     

    {rac-1-[(2-methylpropanoyl)oxy]ethoxy}carbonyl (INNCN)

    estafenatox (INNRG)

     

    glycylglycyl-L-proline (linker) fusion protein with enterotoxin type A (Staphylococcus aureus)-(1-33)-peptidyl-L-seryl[Ser36,Ser37,Glu38,Lys39,Ala41,Thr46,Thr71,Ala72,Ser75,Glu76,Glu78,Ser80,Ser81,Thr214,Ser217,Thr219,Ser220,Ser222,Ser224]enterotoxin type E (Staphylococcus aureus)-(32-230)-peptide (synthetic superantigen SEA/E-120) (INNCN)

    etexilate (INNRG)

     

    ethyl, (hexyloxy)carbonyl

    fosamil (INNRG)

     

    phosphono (INNCN)

    glucuronide (INNRG)

     

    β-D-glucopyranosiduronic acid [oside] (INNCN)

    medocaril (INNRG)

     

    [(5-methyl-2-oxo-1,3-dioxol-4-yl)methoxy]carbonyl (INNCN)

    paptox (INNRG)

     

    protein PAP (Phytolacca americana antiviral) (INNCN)

    placarbil (INNRG)

     

    (R)-2-methyl-1-[(2-methylpropanoyl)oxy]propoxy}carbonyl) (INNCN)

    The systematic name of the following prefix or suffix is amended as follows:

    Preferred prefix or suffix

    Synonym

    Systematic name when different

    aritox (INNRG)

     

    ricin A chain (INNCN)


    ANNEX III

    List of pharmaceutical intermediates, i.e. compounds used for the manufacture of finished pharmaceutical products, to be added to the list of products receiving duty-free treatment included in Annex 6 to Annex I to Regulation (EEC) No 2658/87

    CN code

    CAS RN

    Name

    2843 29 00

    22199-08-2

    [4-amino-N-(pyrimidin-2(1H)-ylidene-κN1)benzenesulfonamidato-κO]silver

    2905 39 95

    281214-27-5

    (2R,3R)-2,3-dimethylbutane-1,4-diyl bis(4-methylbenzenesulfonate)

    2905 59 98

    441002-17-1

    4-chlorobutyl 2-nitrobenzenesulfonate

    2909 30 90

    92878-95-0

    2-(3-chloropropoxy)-1-methoxy-4-nitrobenzene

    2909 30

    503070-57-3

    2-({2-[(6-bromohexyl)oxy]ethoxy}methyl)-1,3-dichlorobenzene

    2909 30

    461432-23-5

    4-(5-bromo-2-chlorobenzyl)phenyl ethyl ether

    2909 49 80

    185954-75-0

    (3R)-3-methoxydecan-1-ol

    2909 49 80

    85309-91-7

    2-[(2,6-dichlorobenzyl)oxy]ethanol

    2909 49 80

    160969-03-9

    2-[2-(2,2,2-trifluoroethoxy)phenoxy]ethyl methanesulfonate

    2909 50 00

    167145-13-3

    2-[2-(3-methoxyphenyl)ethyl]phenol

    2910 20 00

    15448-47-2

    (2R)-2-methyloxirane

    2910 90 00

    62600-71-9

    (2R)-2-(3-chlorophenyl)oxirane

    2910 90 00

    702687-42-1

    (2R)-2-[(5-bromo-2,3-difluorophenoxy)methyl]oxirane

    2910 90 00

    683276-64-4

    [(2R)-2-methyloxiran-2-yl]methyl 4-nitrobenzenesulfonate

    2913 00 00

    90035-34-0

    4′-(trifluoromethyl)biphenyl-4-carbaldehyde

    2914 40 90

    17752-16-8

    (3β)-3-hydroxycholest-5-en-24-one

    2914 50 00

    974-23-2

    (3β,16α)-3-hydroxy-16,17-epoxypregn-5-en-20-one

    2914 70 00

    13054-81-4

    4-chloro-heptane-3,5-dione

    2914 70 00

    10226-30-9

    6-chlorohexan-2-one

    2915 60 90

    53064-79-2

    iodomethyl pivalate

    2915 90 00

    22328-90-1

    (3R)-3-methylhexanoic acid

    2915 90 00

    1069-66-5

    sodium 2-propylpentanoate

    2916 20 00

    211515-46-7

    1-(2-ethylbutyl)cyclohexanecarbonyl chloride

    2916 20 00

    381209-09-2

    1-(2-ethylbutyl)cyclohexanecarboxylic acid

    2916 20 00

    7077-05-6

    trans-4-(propan-2-yl)cyclohexanecarboxylic acid

    2916 39 00

    21900-39-0

    5-fluoro-2-methylbenzoyl chloride

    2916 39 00

    17625-03-5

    sodium hydrogen 3-sulfonatobenzoate

    2917 19 90

    76-72-2

    diethyl ethyl(pentan-2-yl)propanedioate

    2918 29 00

    376592-58-4

    5′-chloro-2′-hydroxy-3′-nitrobiphenyl-3-carboxylic acid

    2918 99 90

    709031-28-7

    (3-hydroxytricyclo[3.3.1.1(3,7)]dec-1-yl)(oxo)acetic acid

    2918 99 90

    35480-52-5

    2,5-bis(2,2,2-trifluoroethoxy)benzoic acid

    2918 99 90

    4651-67-6

    (3α,5β)-3-hydroxy-7-oxocholan-24-oic acid

    2918 99 90

    52179-28-9

    ethyl 2-[4-(2,2-dichlorocyclopropyl)phenoxy]-2-methylpropanoate

    2918 99 90

    530141-60-7

    methyl 3-(5-{[4-(cyclopentyloxy)-2-hydroxyphenyl]carbonyl}-2-hydroxyphenyl)propanoate

    2920 90 10

    91526-18-0

    4-(hydroxymethyl)-5-methyl-1,3-dioxol-2-one

    2921 49 00

    334477-60-0

    (1R)-1-[3,5-bis(trifluoromethyl)phenyl]-N-methylethanamine

    2921 49 00

    376608-71-8

    (1R,2S)-2-(3,4-difluorophenyl)cyclopropanaminium (2R)-hydroxy(phenyl)ethanoate

    2921 49 00

    1034457-07-2

    2-(2,3-dihydro-1H-inden-2-yl)propan-2-amine hydrochloride

    2921 49 00

    945717-05-5

    2-(4-chloro-3-ethylphenyl)ethanamine hydrochloride

    2921 49 00

    89-97-4

    2-chlorobenzylamine

    2921 49 00

    945717-43-1

    N-(4-tert-butylbenzyl)-2-(4-chloro-3-ethylphenyl)ethanamine

    2921 51 90

    150812-21-8

    N4-[(4-fluorophenyl)methyl]-2-nitro-1,4-benzenediamine

    2922 19 85

    1035455-90-3

    (2R)-1-(5-bromo-2,3-difluorophenoxy)-3-{[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]amino}propan-2-ol hydrochloride

    2922 19 85

    0-00-0

    [2-(chloromethyl)-4-(dibenzylamino)phenyl]methanol hydrochloride

    2922 19 85

    133-51-7

    antimonic acid – 1-deoxy-1-(methylamino)-D-glucitol (1:1)

    2922 19 85

    1035455-87-8

    ethyl (2E)-3-(3-{[(2R)-3-{[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]amino}-2-hydroxypropyl]oxy}-4,5-difluorophenyl)prop-2-enoate hydrochloride

    2922 19 85

    702686-97-3

    ethyl 3-(3-{[(2R)-3-{[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]amino}-2-hydroxypropyl]oxy}-4,5-difluorophenyl)propanoate hydrochloride

    2922 29 00

    20059-73-8

    2-[4-(aminomethyl)phenoxy]-N,N-dimethylethanamine

    2922 49 85

    848133-35-7

    (2E)-4-(dimethylamino)but-2-enoic acid hydrochloride

    2922 49 85

    610300-07-7

    (3S,5R)-3-amino-5-methyloctanoic acid

    2922 49 85

    610300-00-0

    (3S,5R)-3-amino-5-methyloctanoic acid hydrochloride

    2922 49 85

    143785-86-8

    4-(1-aminocyclopropyl)-2,3,5-trifluorobenzoic acid

    2922 49 85

    848949-85-9

    4-fluoro-L-leucine – ethyl hydrogen sulfate (1:1)

    2922 49 85

    39068-93-4

    methyl 2-(dimethylamino)-2-phenylbutanoate

    2922 49 85

    168619-25-8

    methyl 3′-aminobiphenyl-3-carboxylate

    2922 49 85

    82834-12-6

    N-[(2S)-1-ethoxy-1-oxopentan-2-yl]-L-alanine

    2922 49 85

    94133-84-3

    sodium 2-amino-2-phenylbutanoate

    2922 50 00

    503070-58-4

    triphenylacetic acid – 4-{(1R)-2-[(6-{2-[(2,6-dichlorobenzyl)oxy]ethoxy}hexyl)amino]-1-hydroxyethyl}-2-(hydroxymethyl)phenol (1:1)

    2924 19 00

    62009-47-6

    2-aminomalonamide

    2924 19 00

    7355-58-0

    N-(2-chloroethyl)acetamide

    2924 29 98

    361442-00-4

    {2-[(tert-butoxycarbonyl)amino]-3-hydroxytricyclo[3.3.1.1(3,7)]dec-1-yl}acetic acid

    2924 29 98

    266993-72-0

    2,3-diaminobenzamide dihydrochloride

    2924 29 98

    168080-49-7

    2-chloro-4-{[(5-fluoro-2-methylphenyl)carbonyl]amino}benzoic acid

    2924 29 98

    317374-08-6

    2-methyl-4-{[(2-methylphenyl)carbonyl]amino}benzoic acid

    2924 29 98

    143785-84-6

    4-(1-carbamoylcyclopropyl)-2,3,5-trifluorobenzoic acid

    2924 29 98

    143785-87-9

    4-[1-(acetylamino)cyclopropyl]-2,3,5-trifluorobenzoic acid

    2924 29 98

    108166-22-9

    4-{[(2-methylphenyl)carbonyl]amino}benzoic acid

    2924 29 98

    150812-23-0

    ethyl {4-[(4-fluorobenzyl)amino]-2-nitrophenyl}carbamate

    2924 29 98

    22316-45-6

    ethyl 3-[(5-chloro-2-nitrophenyl)(phenyl)amino]-3-oxopropanoate

    2924 29 98

    316173-29-2

    methyl (1S,2S,3S,4R)-3-[(1S)-1-amino-2-ethylbutyl]-4-[(tert-butoxycarbonyl)amino]-2-hydroxycyclopentanecarboxylate

    2924 29 98

    1142-20-7

    N-benzyloxycarbonyl-L-alanine

    2924 29 98

    84996-93-0

    N-cyclohexyl-5-hydroxypentanamide

    2924 29 98

    579494-66-9

    propyl {4-[2-(diethylamino)-2-oxoethoxy]-3-ethoxyphenyl}acetate

    2925 19 95

    265136-65-0

    ethyl 3-amino-4-[2-(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)ethoxy]but-2-enoate

    2926 90 95

    855425-38-6

    1-(2-ethylbutyl)cyclohexanecarbonitrile

    2926 90 95

    846023-24-3

    2-cyano-N-(2,4-dichloro-5-methoxyphenyl)acetamide

    2926 90 95

    591769-05-0

    3-cyclopentylprop-2-enenitrile

    2926 90 95

    20099-89-2

    4-(bromoacetyl)benzonitrile

    2926 90 95

    474554-45-5

    4,5-diethoxy-3-fluorobenzene-1,2-dicarbonitrile

    2926 90 95

    79370-78-8

    5-hydroxybenzene-1,3-dicarbonitrile

    2926 90 95

    139481-28-0

    methyl 2-{[(2′-cyanobiphenyl-4-yl)methyl]amino}-3-nitrobenzoate

    2928 00 90

    860035-10-5

    1-({[(2,5-dioxopyrrolidin-1-yl)oxy]carbonyl}oxy)ethyl 2-methylpropanoate

    2928 00 90

    910656-45-0

    2-hydroxy-2-(trifluoromethyl)butanehydrazide

    2928 00 90

    95759-10-7

    4-chloro-2-[(2-methoxy-2-oxoethoxy)imino]-3-oxobutanoic acid

    2928 00 90

    473927-63-8

    ethyl (2Z)-chloro[2-(4-methoxyphenyl)hydrazinylidene]ethanoate

    2928 00 90

    158671-29-5

    N,2-dihydroxy-4-methylbenzamide

    2928 00 90

    84080-68-2

    tert-butyl (2Z)-2-[(2-methoxy-2-oxoethoxy)imino]-3-oxobutanoate

    2928 00 90

    268544-50-9

    tert-butyl-2-[(2-methoxy-2-oxoethoxy)imino]-3-oxobutanoate

    2930 90 99

    13459-62-6

    {2-[(4-chlorophenyl)sulfanyl]phenyl}acetic acid

    2930 90 99

    211513-21-2

    1-(2-ethylbutyl)-N-(2-sulfanylphenyl)cyclohexanecarboxamide

    2930 90 99

    860035-07-0

    1-{[(methylsulfanyl)carbonyl]oxy}ethyl 2-methylpropanoate

    2930 90 99

    893407-18-6

    2,2,2-trifluoro-1-[4′-(methylsulfonyl)biphenyl-4-yl]ethanone

    2930 90 99

    60759-00-4

    3,4-diethoxybenzenecarbothioamide

    2930 90 99

    21048-05-5

    N-methylbenzenecarbothiohydrazide

    2931 00 99

    13682-94-5

    (2-bromoethenyl)(trimethyl)silane

    2931 00 99

    914922-89-7

    (2R,4R)-4-[[(1,1-dimethylethyl)dimethylsilyl]oxy]-N-methoxy-N,2-dimethyl-7-oxoheptanamide

    2931 00 99

    914922-88-6

    (2R,4R)-4-{[tert-butyl(dimethyl)silyl]oxy}-N-methoxy-N,2-dimethyloct-7-enamide

    2931 00 99

    871355-80-5

    (4R)-2-bromo-7-{[tert-butyl(diphenyl)silyl]oxy}hept-1-en-4-yl 4-methylbenzenesulfonate

    2931 00 99

    89694-48-4

    (5-chloro-2-methoxyphenyl)boronic acid

    2931 00 99

    701278-08-2

    [(1R,5S)-5-[dimethyl(phenyl)silyl]-2-{[(2-methoxypropan-2-yl)oxy]methyl}cyclopent-2-en-1-yl]methanol

    2931 00 99

    701278-09-3

    {(4S,5R)-5-[(benzyloxy)methyl]-4-[dimethyl(phenyl)silyl]cyclopent-1-en-1-yl}methanol

    2931 00 99

    796967-18-5

    1-(2-fluoro-5-methylphenyl)-3-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]urea

    2931 00 99

    172732-52-4

    2-(1,3,2-dioxaborinan-2-yl)benzonitrile

    2931 00 99

    185411-12-5

    methyl 3-(trimethylsilyl)pent-4-enoate

    2932 19 00

    253128-10-8

    (1S)-1,5:7,10-dianhydro-12,13-bis-O-[tert-butyl(dimethyl)silyl]-2,3,4,6,8,11-hexadeoxy-1-{2-[(2S,5S)-5-(3-hydroxypropyl)-3-methylidenetetrahydrofuran-2-yl]ethyl}-3-methyl-9-O-methyl-4-methylidene-8-[(phenylsulfonyl)methyl]-D-arabino-D-altro-tridecitol

    2932 19 00

    441045-17-6

    (1S,3S,6S,9S,12S,14R,16R,18S,20R,21R,22S,26R,29S,31R,32S,33R,35R,36S)-20-[(2S)-3-amino-2-hydroxypropyl]-21-methoxy-14-methyl-8,15-bis(methylene)-2,19,30,34,37,39,40,41-octaoxanonacyclo[24.9.2.13,32.13,33.16,9.112,16.018,22.029,36.031,35]hentetracontan-24-one methanesulfonate

    2932 29 85

    916069-80-2

    (4S)-4-(fluoromethyl)dihydrofuran-2(3H)-one

    2932 29 85

    63106-93-4

    1-phenyl-3-oxabicyclo[3.1.0]hexan-2-one

    2932 29 85

    7734-80-7

    2-oxo-2H-chromene-6-carboxylic acid

    2932 29 85

    0-00-0

    4-(4-fluorophenyl)-7-(isothiocyanatomethyl)-2H-chromen-2-one

    2932 29 85

    947408-91-5

    6-[(2,4-dihydroxyphenyl)carbonyl]-2H-chromen-2-one

    2932 29 85

    947408-90-4

    6-[(2,4-dimethoxyphenyl)carbonyl]-2H-chromen-2-one

    2932 99 00

    452342-08-4

    (1R)-2-(benzylamino)-1-(2,2-dimethyl-4H-1,3-benzodioxin-6-yl)ethanol

    2932 99 00

    99541-23-8

    (1R,2S,3R,4R,5R)-4-azido-2-{[(4aR,6S,7R,8S,8aR)-7,8-bis(benzyloxy)-2-phenylhexahydropyrano[3,2-d][1,3]dioxin-6-yl]oxy}-6,8-dioxabicyclo[3.2.1]oct-3-yl acetate

    2932 99 00

    461432-25-7

    (1S)-2,3,4,6-tetra-O-acetyl-1,5-anhydro-1-[4-chloro-3-(4-ethoxybenzyl)phenyl]-D-glucitol

    2932 99 00

    196597-79-2

    (2E)-1,2,6,7-tetrahydro-8H-indeno[5,4-b]furan-8-ylideneethanenitrile

    2932 99 00

    3308-94-9

    2-(3-chloropropyl)-2-(4-fluorophenyl)-1,3-dioxolane

    2932 99 00

    274693-53-7

    [(3aS,4R,6S,6aR)-6-hydroxy-2,2-dimethyltetrahydro-3aH-cyclopenta[d][1,3]dioxol-4-yl]carbamate

    2932 99 00

    185954-98-7

    [6(2Z,3R)]-3-O-decyl-2-deoxy-6-O-[2-deoxy-3-O-(3-metoxydecyl)-6-methyl-2-[(1-oxo-11-octadecenyl)amino]-4-O-phosphono-β-D-glucopyranosyl]-2-[(1,3-dioxotetradecyl)amino]-α-D-glucopyranose 1-(dihydrogen phosphate) tetrasodium salt

    2932 99 00

    136172-58-2

    1,6-di-O-acetyl-2-azido-3,4-di-O-benzyl-2-deoxy-D-glucopyranose

    2932 99 00

    196597-80-5

    2-[(8S)-1,6,7,8-tetrahydro-2H-indeno[5,4-b]furan-8-yl]ethanamine hydrochloride

    2932 99 00

    666860-59-9

    2-amino-2-oxoethyl{3-[trans-5-(6-methoxynaphthalen-1-yl)-1,3-dioxan-2-yl]propyl}carbamate

    2932 99 00

    117661-72-0

    5-(chloromethyl)-6-methyl-1,3-benzodioxole

    2932 99 00

    959624-24-9

    6-(hydroxymethyl)-4-phenyl-3,4-dihydro-2H-chromen-2-ol

    2932 99 00

    960404-59-5

    but-2-yne-1,4-diol – methyl 1-C-[4-chloro-3-(4-ethoxybenzyl)phenyl]-α-D-glucopyranoside (1:1)

    2932 99 00

    15826-37-6

    disodium 5,5′-[(2-hydroxypropane-1,3-diyl)bis(oxy)]bis(4-oxo-4H-chromene-2-carboxylate)

    2932 99 00

    204254-84-2

    ethyl (3aR,7R,7aR)-2,2-dimethyl-7-[(methylsulfonyl)oxy]-3a,6,7,7a-tetrahydro-1,3-benzodioxole-5-carboxylate

    2932 99 00

    99541-26-1

    methyl (2S,3S,4S,5S,6S)-6-{[(1S,2S,3S,4R,5R)-3-(acetyloxy)-4-azido-6,8-dioxabicyclo[3.2.1]oct-2-yl]methyl}-4,5-bis(benzyloxy)-3-hydroxytetrahydro-2H-pyran-2-carboxylate

    2932 99 00

    114869-97-5

    methyl 6-O-acetyl-4-O-(2-O-acetyl-3-O-benzyl-6-methyl-α-L-idopyranuronosyl)-3-O-benzyl-2-{[(benzyloxy)carbonyl]amino}-2-deoxy-α-D-glucopyranoside

    2933 19 90

    1035677-60-1

    (4S)-3-(4-chlorophenyl)-N-methyl-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboximidamide 2,3-dihydroxybutanedioate

    2933 19 90

    18048-64-1

    2-(3,4-dimethylphenyl)-5-methyl-2,4-dihydro-3H-pyrazol-3-one

    2933 19 90

    1035675-24-1

    3-(4-chlorophenyl)-N-methyl-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboximidamide

    2933 19 90

    1028026-83-6

    5-methyl-1-(propan-2-yl)-4-[4-(propan-2-yloxy)benzyl]-1,2-dihydro-3H-pyrazol-3-one

    2933 19 90

    473921-12-9

    5-{[3,5-diethyl-1-(2-hydroxyethyl)-1H-pyrazol-4-yl]oxy}benzene-1,3-dicarbonitrile

    2933 29 90

    65902-59-2

    2-bromo-4-nitro-1H-imidazole

    2933 29 90

    57531-37-0

    2-chloro-4-nitro-1H-imidazole

    2933 29 90

    1000164-35-1

    3-(1,1-dimethylethyl)-N-[(9H-fluoren-9-ylmethoxy)carbonyl]-1-(triphenylmethyl)-L-histidyl-2-methylalanyl-L-α-glutamylglycine

    2933 29 90

    152074-97-0

    L-α-aspartyl-L-α-glutamyl-L-asparaginyl-L-prolyl-L-valyl-L-valyl-L-histidyl-L-phenylalanyl-L-phenylalanyl-L-lysyl-L-asparaginyl-L-isoleucyl-L-valyl-L-threonyl-L-prolyl-L-arginyl-L-threonine

    2933 29 90

    781666-30-6

    L-α-aspartyl-L-α-glutamyl-L-asparaginyl-L-prolyl-L-valyl-L-valyl-L-histidyl-L-phenylalanyl-L-phenylalanyl-L-lysyl-L-asparaginyl-L-isoleucyl-L-valyl-L-threonyl-L-prolyl-L-arginyl-L-threonine tetraacetate

    2933 29 90

    451470-33-0

    methyl 3′-(2-methyl-4,5-dihydro-1H-imidazol-1-yl)biphenyl-3-carboxylate

    2933 39 99

    925978-49-0

    (+)-5-[6-(1-methyl-1H-pyrazol-4-yl)pyridin-3-yl]-1-azabicyclo[3.2.1]octane

    2933 39 99

    876170-44-4

    (1S,5S)-3-(5,6-dichloropyridin-3-yl)-3,6-diazabicyclo[3.2.0]heptane benzenesulfonate

    2933 39 99

    741705-70-4

    (2R)-phenyl[(2R)-piperidin-2-yl]ethanoic acid hydrochloride

    2933 39 99

    414910-13-7

    (2S)-hydroxy(phenyl)ethanoic acid – (2R)-2-(4-fluoro-2-methylphenyl)piperidin-4-one (1:1)

    2933 39 99

    0-00-0

    (3aR,6aR)-1-(pyridin-3-yl)octahydropyrrolo[3,4-b]pyrrole 4-methylbenzenesulfonate

    2933 39 99

    370882-57-8

    (3aR,6aR)-1-(pyridin-3-yl)octahydropyrrolo[3,4-b]pyrrole dihydrochloride

    2933 39 99

    334618-23-4

    (3R)-piperidin-3-amine dihydrochloride

    2933 39 99

    1062580-52-2

    (3R,4R)-1-benzyl-N,4-dimethylpiperidin-3-amine dihydrochloride

    2933 39 99

    27262-47-1

    (S)-1-butyl-N-(2,6-dimethylphenyl)piperidine-2-carboxamide

    2933 39 99

    105812-81-5

    [(3S,4R)-4-(4-fluorophenyl)-1-methylpiperidin-3-yl]methanol

    2933 39 99

    876068-51-8

    [(3S,4S)-4-amino-1-(5,6-dichloropyridin-3-yl)pyrrolidin-3-yl]methanol

    2933 39 99

    871022-14-9

    1-({4-[({[2-oxo-3-(propan-2-yl)-2,3-dihydro-1H-benzimidazol-1-yl]carbonyl}amino)methyl]piperidin-1-yl}methyl)cyclobutanecarboxylic acid

    2933 39 99

    5421-92-1

    1-(pyridin-4-yl)pyridinium chloride hydrochloride

    2933 39 99

    272776-12-2

    1,1′-binaphthalene-2,2′-diol –5-methoxy-2-{(S)-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]sulfinyl}-1H-benzimidazole (1:1)

    2933 39 99

    871022-19-4

    1-[(4-{[(tert-butoxycarbonyl)amino]methyl}piperidin-1-yl)methyl]cyclobutanecarboxylic acid

    2933 39 99

    3613-73-8

    2,8-dimethyl-5-[2-(6-methylpyridin-3-yl)ethyl]-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole

    2933 39 99

    179687-79-7

    2-[(2-chloro-4-nitrophenoxy)methyl]pyridine

    2933 39 99

    122321-04-4

    2-[methyl(pyridin-2-yl)amino]ethanol

    2933 39 99

    945405-37-8

    2-methyl-3-[(2S)-pyrrolidin-2-ylmethoxy]pyridine 2,3-dihydroxybutanedioate

    2933 39 99

    936637-40-0

    3,3′-piperidine-1,4-diyldipropan-1-ol 4-methylbenzenesulfonate

    2933 39 99

    88150-62-3

    3-ethyl-5-methyl-4-(2-chlorophenyl)-2-{[2-(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)ethoxy]methyl}-6-methyl-1,4-dihydropyridine-3,5-dicarboxylate

    2933 39 99

    84100-54-9

    4-(ethylamino)piperidine-4-carboxamide

    2933 39 99

    873546-30-6

    4,4′-[piperidine-1,4-diylbis(propane-3,1-diyloxy)]bis(N′-hydroxybenzenecarboximidamide)

    2933 39 99

    873546-74-8

    4,4′-[piperidine-1,4-diylbis(propane-3,1-diyloxy)]bis[N′-(acetyloxy)benzenecarboximidamide]

    2933 39 99

    873546-38-4

    4,4′-[piperidine-1,4-diylbis(propane-3,1-diyloxy)]dibenzenecarboximidamide trihydrochloride pentahydrate

    2933 39 99

    873546-80-6

    4,4′-[piperidine-1,4-diylbis(propane-3,1-diyloxy)]dibenzonitrile

    2933 39 99

    78750-61-5

    4-[(3-nitropyridin-2-yl)amino]phenol

    2933 39 99

    866109-93-5

    4-{4-[4-(trifluoromethoxy)phenoxy]piperidin-1-yl}phenol 4-methylbenzenesulfonate

    2933 39 99

    927889-51-8

    4-bromo-2,6-diethylpyridine 4-methylbenzenesulfonate

    2933 39 99

    691882-47-0

    4-hydroxybenzoic acid – (2S,4E)-N-methyl-5-[5-(propan-2-yloxy)pyridin-3-yl]pent-4-en-2-amine (1:1)

    2933 39 99

    876068-46-1

    5,6-dichloro-N-(2,2-dimethoxyethyl)pyridin-3-amine

    2933 39 99

    1072-98-6

    5-chloropyridin-2-amine

    2933 39 99

    298692-34-9

    6-(chloroacetyl)pyridine-2-carboxylic acid

    2933 39 99

    550349-58-1

    7-chloro-3-(6-methoxypyridin-3-yl)-N,N,5-trimethyl-4-oxo-4,5-dihydro-3H-pyridazino[4,5-b]indole-1-carboxamide

    2933 39 99

    414909-98-1

    benzyl 2-(4-fluoro-2-methylphenyl)-4-oxo-3,4-dihydropyridine-1(2H)-carboxylate

    2933 39 99

    56880-11-6

    ethyl [(3-endo)-8-methyl-8-azabicyclo[3.2.1]oct-3-yl)acetate

    2933 39 99

    548797-97-3

    N-(2-{[(2S)-3-{[1-(4-chlorobenzyl)piperidin-4-yl]amino}-2-hydroxy-2-methylpropyl]oxy}-4-hydroxyphenyl)acetamide

    2933 39 99

    0-00-0

    N-[(S)-1-azabicyclo[2.2.2]oct-2-yl(phenyl)methyl]-2,6-dichloro-3-(trifluoromethyl)benzamide hydrochloride

    2933 39 99

    329003-65-8

    sodium hydrogen [1-hydroxy-1-phosphono-2-(pyridin-3-yl)ethyl]phosphonate hemipentahydrate

    2933 49 10

    417716-92-8

    4-{3-chloro-4-[(cyclopropylcarbamoyl)amino]phenoxy}-7-methoxyquinoline-6-carboxamide methanesulfonate

    2933 49 90

    503291-53-0

    2-ethylbutyl (3S,4aS,6S,8aR)-6-[3-chloro-2-(1H-tetrazol-5-yl)phenoxy]decahydro-3-isoquinolinecarboxylate 4-methylbenzenesulfonate

    2933 49 90

    103733-32-0

    benzyl (3S)-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-3-carboxylate hydrochloride

    2933 49 90

    503293-98-9

    (3S,4aS,6S,8aR)-6-hydroxy-2-(methoxycarbonyl)decahydroisoquinoline-3-carboxylic acid

    2933 49 90

    503290-66-2

    (3S,4aS,6S,8aR)-6-[3-chloro-2-(2H-tetrazol-5-yl)phenoxy]decahydro-3-isoquinolinecarboxylic acid hydrochloride

    2933 49 90

    134388-95-7

    (3S,4aS,8aR)-2-(methoxycarbonyl)-6-oxodecahydroisoquinoline-3-carboxylic acid – (1R)-1-phenylethanamine (1:1)

    2933 49 90

    868210-14-4

    4-(4-{[(2S,4R)-4-[acetyl(4-chlorophenyl)amino]-2-methyl-3,4-dihydroquinolin-1(2H)-yl]carbonyl}phenoxy)-2,2-dimethylbutanoic acid

    2933 49 90

    00-00-0

    methyl 2-[(3R)-3-{3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]phenyl}-3-({[1-(hydroxymethyl)cyclopropyl]methyl}sulfanyl)propyl]benzoate hydrochloride

    2933 49 90

    848133-76-6

    N-(4-chloro-3-cyano-7-ethoxyquinolin-6-yl)acetamide

    2933 59 95

    869490-23-3

    (3,3-difluoropyrrolidin-1-yl){(2S,4S)-4-[4-(pyrimidin-2-yl)piperazin-1-yl]pyrrolidin-2-yl}methanone

    2933 59 95

    941685-40-1

    (3R)-3-cyclopentyl-3-[4-(7-{[2-(trimethylsilyl)ethoxy]methyl}-7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]propanenitrile

    2933 59 95

    941678-49-5

    (3R)-3-cyclopentyl-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]propanenitrile

    2933 59 95

    941685-41-2

    (3S)-3-cyclopentyl-3-[4-(7-{[2-(trimethylsilyl)ethoxy]methyl}-7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]propanenitrile

    2933 59 95

    957187-34-7

    [(8R)-8-(3,5-difluorophenyl)-10-oxo-6,9-diazaspiro[4.5]dec-9-yl]acetic acid

    2933 59 95

    356058-42-9

    {2-[(4-fluorobenzyl)sulfanyl]-4-oxo-4,5,6,7-tetrahydro-1H-cyclopenta[d]pyrimidin-1-yl}acetic acid

    2933 59 95

    0-00-0

    2,3-dihydroxy-2,3-bis(phenylcarbonyl)butanedioic acid – ethyl [(8R)-8-(3,5-difluorophenyl)-10-oxo-6,9-diazaspiro[4.5]dec-9-yl]acetate (1:1)

    2933 59 95

    90213-66-4

    2,4-dichloro-7H-pyrrolo[2,3-d]pyrimidine

    2933 59 95

    3934-20-1

    2,4-dichloropyrimidine

    2933 59 95

    451487-18-6

    2-[(4-fluorobenzyl)sulfanyl]-1,5,6,7-tetrahydro-4H-cyclopenta[d]pyrimidin-4-one

    2933 59 95

    865758-96-9

    2-[(6-chloro-3-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)methyl]benzonitrile

    2933 59 95

    934815-71-1

    2-[3-(6-{[2-(2,4-dichlorophenyl)ethyl]amino}-2-methoxypyrimidin-4-yl)phenyl]-2-methylpropanoic acid phosphate

    2933 59 95

    722543-31-9

    2-{ethyl[3-({4-[(5-{2-[(3-fluorophenyl)amino]-2-oxoethyl}-1H-pyrazol-3-yl)amino]quinazolin-7-yl}oxy)propyl]amino}ethyl dihydrogen phosphate

    2933 59 95

    1032066-96-8

    2-amino-9-{(1S,3R,4S)-3-[(benzyloxy)methyl]-4-[dimethyl(phenyl)silyl]-2-methylidenecyclopentyl}-1,9-dihydro-6H-purin-6-one – methanesulfonate (2:1)

    2933 59 95

    540737-29-9

    3-{(3R,4R)-4-methyl-3-[methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrile 2-hydroxypropane-1,2,3-tricarboxylate

    2933 59 95

    1137917-12-4

    3-{[6-(ethylsulfonyl)pyridin-3-yl]oxy}-5-{[(2S)-1-hydroxypropan-2-yl]oxy}benzoic acid – 1,4-diazabicyclo[2.2.2]octane (2:1)

    2933 59 95

    941685-39-8

    3-cyclopentyl-3-[4-(7-{[2-(trimethylsilyl)ethoxy]methyl}-7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]propanenitrile

    2933 59 95

    941685-27-4

    4-(1H-pyrazol-4-yl)-7-{[2-(trimethylsilyl)ethoxy]methyl}-7H-pyrrolo[2,3-d]pyrimidine

    2933 59 95

    1780-26-3

    4,6-dichloro-2-methylpyrimidine

    2933 59 95

    145783-14-8

    4,6-dichloro-5-nitro-2-(propylsulfanyl)pyrimidine

    2933 59 95

    3680-69-1

    4-chloro-7H-pyrrolo[2,3-d]pyrimidine

    2933 59 95

    61379-64-4

    4-cyclopentylpiperazin-1-amine

    2933 59 95

    55112-42-0

    4-methylpiperazine-1-carbonyl chloride hydrochloride

    2933 59 95

    0-00-0

    5-(benzylamino)-2-(3-methoxyphenyl)-7-(4-methylpiperazin-1-yl)[1,2,4]triazolo[1,5-a]quinoline-4-carbonitrile – (2E)-but-2-enedioate (2:1) hydrate

    2933 59 95

    55293-96-4

    5,7-dimethyl[1,2,4]triazolo[1,5-a]pyrimidine-2-carbaldehyde

    2933 59 95

    179688-01-8

    7-(benzyloxy)-6-methoxyquinazolin-4(3H)-one

    2933 59 95

    444731-74-2

    N-(2-chloropyrimidin-4-yl)-2,3-dimethyl-2H-indazol-6-amine

    2933 59 95

    0-00-0

    N-(5-fluoro-3-methyl-1H-indol-1-yl)-4-methyl-2-(pyridin-2-yl)pyrimidine-5-carboxamide

    2933 79 00

    586414-48-4

    (-)-3-{3-bromo-4-[(2,4-difluorobenzyl)oxy]-6-methyl-2-oxopyridin-1(2H)-yl}-N,4-dimethylbenzamide

    2933 79 00

    425663-71-4

    (1S)-1-amino-3-methyl-1,3,4,5-tetrahydro-2H-3-benzazepin-2-one hydrochloride

    2933 79 00

    813452-14-1

    (4S)-1-[(2S,3S,11bS)-2-amino-9,10-dimethoxy-1,3,4,6,7,11b-hexahydro-2H-pyrido[2,1-a]isoquinolin-3-yl]-4-(fluoromethyl)pyrrolidin-2-one dihydrochloride

    2933 79 00

    5162-90-3

    3-(2-oxo-1,2-dihydroquinolin-4-yl)alanine

    2933 79 00

    536760-29-9

    3-chloro-1-(4-nitrophenyl)-5,6-dihydropyridin-2(1H)-one

    2933 79 00

    4876-10-2

    4-(bromomethyl)quinolin-2(1H)-one

    2933 79 00

    5057-12-5

    4,6,7,8-tetrahydroquinoline-2,5(1H,3H)-dione

    2933 79 00

    54197-66-9

    6-hydroxy-3,4-dihydroquinolin-2(1H)-one

    2933 79 00

    22246-18-0

    7-hydroxy-3,4-dihydroquinolin-2(1H)-one

    2933 79 00

    536759-91-8

    ethyl 1-(4-methoxyphenyl)-6-(4-nitrophenyl)-7-oxo-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylate

    2933 79 00

    503614-91-3

    ethyl 1-(4-methoxyphenyl)-7-oxo-6-[4-(2-oxopiperidin-1-yl)phenyl]-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylate

    2933 79 00

    586379-61-5

    methyl 3-(4-hydroxy-6-methyl-2-oxopyridin-1(2H)-yl)-4-methylbenzoate

    2933 99 80

    709031-45-8

    (1S,3S,5S)-2-azabicyclo[3.1.0]hexane-3-carboxamide methanesulfonate

    2933 99 80

    649735-46-6

    (2R)-1-({4-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yl}oxy)propan-2-ol

    2933 99 80

    51077-14-6

    (2S)-1-(tert-butoxycarbonyl)azetidine-2-carboxylic acid

    2933 99 80

    631916-97-7

    (2S)-N-{4-[(Z)-amino(methoxyimino)methyl]benzyl}-1-{(2R)-2-[3-chloro-5-(difluoromethoxy)phenyl]-2-hydroxyethanoyl}azetidine-2-carboxamide – benzenesulphonic acid (1:1)

    2933 99 80

    80875-98-5

    (2S,3aS,7aS)-octahydro-1H-indole-2-carboxylic acid

    2933 99 80

    948846-40-0

    (2S,3S)-2,3-bis[(phenylcarbonyl)oxy]butanedioic acid – ethyl (3aR,6aR)-hexahydropyrrolo[3,4-b]pyrrole-5(1H)-carboxylate (1:1)

    2933 99 80

    1000164-36-2

    (5S,8S,11S,14S,17S,20S,23S,26S,29S,32S,35S,38S)-5-(3-amino-3-oxopropyl)-20-benzyl-23-[(2S)-butan-2-yl]-14,38-bis{4-[(tert-butoxycarbonyl)amino]butyl}-29-{[1-(tert-butoxycarbonyl)-1H-indol-3-yl]methyl}-17-(3-tert-butoxy-3-oxopropyl)-1-(1H-fluoren-9-yl)-8,11,26,41,41-pentamethyl-32-(2-methylpropyl)-3,6,9,12,15,18,21,24,27,30,33,36,39-tridecaoxo-35-(propan-2-yl)-2-oxa-4,7,10,13,16,19,22,25,28,31,34,37,40-tridecaazadotetracontan-42-oic acid

    2933 99 80

    22162-51-2

    1-(2-nitrobenzyl)-1H-pyrrole-2-carbaldehyde

    2933 99 80

    35681-40-4

    1-(propan-2-yl)-1,3-dihydro-2H-benzimidazol-2-one

    2933 99 80

    166170-15-6

    1-(tert-butoxycarbonyl)-2-methyl-D-proline

    2933 99 80

    796967-16-3

    1-[4-(3-amino-1H-indazol-4-yl)phenyl]-3-(2-fluoro-5-methylphenyl)urea

    2933 99 80

    0-00-0

    1-[4-(3-amino-1H-indazol-4-yl)phenyl]-3-(2-fluoro-5-methylphenyl)urea hydrochloride

    2933 99 80

    444731-72-0

    2,3-dimethyl-2H-indazol-6-amine

    2933 99 80

    19686-05-6

    2,8-dimethyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole

    2933 99 80

    912444-00-9

    2-[(2R)-2-methylpyrrolidin-2-yl]-1H-benzimidazole-4-carboxamide

    2933 99 80

    912445-36-4

    2-[(2S)-2-methylpyrrolidin-2-yl]-1H-benzimidazole-4-carboxamide dihydrochloride

    2933 99 80

    163457-23-6

    3,3-difluoropyrrolidine hydrochloride

    2933 99 80

    239463-85-5

    3-{5-[(2R)-2-aminopropyl]-7-cyano-2,3-dihydro-1H-indol-1-yl}propyl benzoate (2R,3R)-2,3-dihydroxybutanedioate

    2933 99 80

    55321-99-8

    3-oxo-3,4-dihydropyrazine-2-carboxamide

    2933 99 80

    952490-01-6

    4-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yl 2,2-dimethylpropanoate

    2933 99 80

    942436-93-3

    4-amino-8-(2,5-dimethoxyphenyl)-N-propylcinnoline-3-carboxamide

    2933 99 80

    942437-37-8

    4-amino-8-(2-fluoro-6-methoxyphenyl)-N-propylcinnoline-3-carboxamide

    2933 99 80

    288385-88-6

    4-fluoro-2-methyl-1H-indol-5-ol

    2933 99 80

    503293-47-8

    5-(2-chloro-6-fluorophenyl)-2H-tetrazole

    2933 99 80

    73963-42-5

    5-(4-chlorobutyl)-1-cyclohexyl-1H-tetrazole

    2933 99 80

    606143-52-6

    5-[(4-bromo-2-chlorophenyl)amino]-4-fluoro-N-(2-hydroxyethoxy)-1-methyl-1H-benzimidazole-6-carboxamide

    2933 99 80

    0-00-0

    5-fluoro-1-(3-fluorobenzyl)-N-(1H-indol-5-yl)-1H-indole-2-carboxamide

    2933 99 80

    872206-47-8

    5-methyl-4-oxo-1,4-dihydropyrrolo[2,1-f][1,2,4]triazin-6-yl 2,2-dimethylpropanoate

    2933 99 80

    259793-88-9

    6-bromo-3-oxo-3,4-dihydropyrazine-2-carboxamide

    2933 99 80

    1137606-74-6

    6-fluoro-3-oxo-3,4-dihydropyrazine-2-carbonitrile – N-cyclohexylcyclohexanamine (1:1)

    2933 99 80

    261953-36-0

    6-iodo-1H-indazole

    2933 99 80

    80076-47-7

    8,9-difluoro-5-methyl-1-oxo-6,7-dihydro-1H,5H-pyrido[3,2,1-ij]quinoline-2-carboxylic acid

    2933 99 80

    52602-39-8

    9H-carbazol-4-ol

    2933 99 80

    145641-35-6

    benzyl (2S,3aR,7aS)-octahydro-1H-indole-2-carboxylate hydrochloride

    2933 99 80

    87269-87-2

    benzyl (2S,3aS,6aS)-octahydrocyclopenta[b]pyrrole-2-carboxylate hydrochloride

    2933 99 80

    1012065-72-3

    ethyl 2-amino-9,10-dimethoxy-1,6,7,11b-tetrahydro-4H-pyrido[2,1-a]isoquinoline-3-carboxylate

    2933 99 80

    131707-24-9

    ethyl 6-bromo-5-hydroxy-1-methyl-2-[(phenylsulfanyl)methyl]-1H-indole-3-carboxylate

    2933 99 80

    105152-95-2

    ethyl 7-(3-aminopyrrolidin-1-yl)-1-(2,4-difluorophenyl)-6-fluoro-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxylate

    2933 99 80

    139481-44-0

    methyl 1-[(2′-cyanobiphenyl-4-yl)methyl]-2-ethoxy-1H-benzimidazole-7-carboxylate

    2933 99 80

    0-00-0

    methyl 1-tert-butyl-2-hydroxy-1H-pyrrolo[2,3-b]pyridine-3-carboxylate

    2933 99 80

    21688-11-9

    N2-[(benzyloxy)carbonyl]-L-glutaminyl-L-asparaginyl-S-benzyl-L-cysteinyl-L-prolyl-L-leucylglycinamide

    2933 99 80

    361440-67-7

    tert-butyl (1S,3S,5S)-3-carbamoyl-2-azabicyclo[3.1.0]hexane-2-carboxylate

    2933 99 80

    709031-38-9

    tert-butyl (2S)-2-carbamoyl-2,3-dihydro-1H-pyrrole-1-carboxylate

    2933 99 80

    709031-43-6

    tert-butyl [(1S)-2-[(1S,3S,5S)-3-cyano-2-azabicyclo[3.1.0]hex-2-yl]-1-(3-hydroxytricyclo[3.3.1.1(3,7)]dec-1-yl)-2-oxoethyl]carbamate

    2933 49 90

    936359-25-0

    methyl 2-((R)-3-(3-((E)-2-(7-chloroquinolin-2-yl)vinyl)phenyl)-3-(((1-(hydroxymethyl)cyclopropyl)methyl)sulfanyl)propyl)benzoate

    2934 10 00

    110130-88-6

    (2Z)-[(acetyloxy)imino](2-amino-1,3-thiazol-4-yl)ethanoic acid

    2934 10 00

    68672-66-2

    (2Z)-{[(1-tert-butoxy-2-methyl-1-oxopropan-2-yl)oxy]imino}[2-(tritylamino)-1,3-thiazol-4-yl]ethanoic acid

    2934 10 00

    291536-35-1

    (5Z)-5-(4-fluorobenzylidene)-1,3-thiazolidine-2,4-dione

    2934 10 00

    302964-24-5

    2-amino-N-(2-chloro-6-methylphenyl)-1,3-thiazole-5-carboxamide

    2934 10 00

    866920-24-3

    3-[2-chloro-4-({4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}methoxy)phenyl]-1,2,4-oxadiazol-5(4H)-one

    2934 10 00

    752253-39-7

    4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl]-5-methyl-N-(prop-2-yn-1-yl)-1,3-thiazol-2-amine

    2934 10 00

    914361-45-8

    L-lysine – {[(2R,3R)-3-[4-(4-cyanophenyl)-1,3-thiazol-2-yl]-2-(2,4-difluorophenyl)-1-(1H-1,2,4-triazol-1-yl)butan-2-yl]oxy}methyl dihydrogen phosphate – ethanol (1:1:1)

    2934 10 00

    302964-08-5

    N-(2-chloro-6-methylphenyl)-2-[(6-chloro-2-methylpyrimidin-4-yl)amino]-1,3-thiazole-5-carboxamide

    2934 10 00

    127660-04-2

    sodium (2Z)-(2-amino-1,3-thiazol-4-yl)(hydroxyimino)ethanoate

    2934 99 90

    17381-54-3

    (1-benzothiophen-5-yl)acetic acid

    2934 99 90

    630100-90-2

    (1R)-1,2-anhydro-4-C-{(1E,3E)-4-[(1S,2S,3E,5R,6R,9R)-5-(1-carboxylato-4-cycloheptylpiperazin-2-yl)-6,9-dihydroxy-2,6-dimethyl-11-oxooxacyclododec-3-en-1-yl]penta-1,3-dien-1-yl}-3,5-dideoxy-1-[(2R,3S)-3-hydroxypentan-2-yl]-D-erythropentitol

    2934 99 90

    220099-91-2

    (2R)-3′H-spiro[4-azabicyclo[2.2.2]octane-2,2′-furo[2,3-b]pyridine]

    2934 99 90

    220100-81-2

    (2R)-3′H-spiro[4-azabicyclo[2.2.2]octane-2,2′-furo[2,3-b]pyridine] (S,S)-2,3-dihydroxybutanedioate

    2934 99 90

    161599-46-8

    (2R,3R,4R,5R)-2-(4-amino-5-fluoro-2-oxopyrimidin-1(2H)-yl)-2-fluoro-5-methyltetrahydrofuran-3,4-diyl diacetate

    2934 99 90

    690270-65-6

    (2R,3S,4R)-5-(4-amino-2-oxopyrimidin-1(2H)-yl)-2-azido-2-{[(2-methylpropanoyl)oxy]methyl}tetrahydrofuran-3,4-diyl bis(2-methylpropanoate) hydrochloride

    2934 99 90

    265121-04-8

    (3-{[(2R,3S)-2-{(1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethoxy}-3-(2-fluorophenyl)morpholin-4-yl]methyl}-5-oxo-2,5-dihydro-1H-1,2,4-triazol-1-yl)phosphonic acid – 1-deoxy-1-(methylamino)-D-glucitol (1:2)

    2934 99 90

    163680-80-6

    (3S)-10-[1-(acetylamino)cyclopropyl]-9-fluoro-3-methyl-7-oxo-2,3-dihydro-7H-[1,4]oxazino[2,3,4-ij]quinoline-6-carboxylic acid

    2934 99 90

    132335-46-7

    (3S)-N,N-dimethyl-3-(naphthalen-1-yloxy)-3-(thiophen-2-yl)propan-1-amine

    2934 99 90

    133413-70-4

    (3S,6R,9S,12R,15S,18R,21S,24R)-6,18-dibenzyl-4,10,12,16,22,24-hexamethyl-3,9,15,21-tetrakis(2-methylpropyl)-1,7,13,19-tetraoxa-4,10,16,22-tetraazacyclotetracosane-2,5,8,11,14,17,20,23-octone

    2934 99 90

    503068-36-8

    (5R)-3-(6-{2-[(2,6-dichlorobenzyl)oxy]ethoxy}hexyl)-5-(2,2-dimethyl-4H-1,3-benzodioxin-6-yl)-1,3-oxazolidin-2-one

    2934 99 90

    452339-73-0

    (5R)-5-(2,2-dimethyl-4H-1,3-benzodioxin-6-yl)-1,3-oxazolidin-2-one

    2934 99 90

    877130-28-4

    (6R)-6-cyclopentyl-6-[2-(2,6-diethylpyridin-4-yl)ethyl]-3-[(5,7-dimethyl[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)methyl]-4-hydroxy-5,6-dihydro-2H-pyran-2-one

    2934 99 90

    132335-44-5

    (S)-3-(dimethylamino)-1-(thiophen-2-yl)propan-1-ol

    2934 99 90

    812647-80-6

    {(2R,3S,4R,5R)-2-azido-5-(2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)-3,4-bis[(phenylcarbonyl)oxy]tetrahydrofuran-2-yl}methyl 3-chlorobenzoate

    2934 99 90

    00-00-0

    1-(1-{4-[2-(4-fluorophenyl)-1,3-dioxolan-2-yl]butyl}-1,2,3,6-tetrahydropyridin-4-yl)-1,3-dihydro-2H-benzimidazol-2-one

    2934 99 90

    1029716-44-6

    1-(1-ethoxyethyl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole

    2934 99 90

    165172-60-1

    1-[(2R,5S)-5-(hydroxymethyl)-2,5-dihydrofuran-2-yl]-5-methylpyrimidine-2,4(1H,3H)-dione – 1-methylpyrrolidin-2-one (1:1)

    2934 99 90

    519187-97-4

    1-[3-(2-benzo[b]thien-5-ylethoxy)propyl]-3-azetidinol – (2Z)-2-butenedioate (1:1)

    2934 99 90

    127000-90-2

    1-{[(2R,3S)-2-(2,4-difluorophenyl)-3-methyloxiran-2-yl]methyl}-1H-1,2,4-triazole

    2934 99 90

    710281-33-7

    2-({[(1R,3S)-3-{[2-(3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}cyclohexyl]oxy}methyl)-6-methylbenzoic acid

    2934 99 90

    96803-30-4

    2-(1-benzothiophen-5-yl)ethanol

    2934 99 90

    913695-00-8

    2-[({4-[(2,2-dimethyl-1,3-dioxan-5-yl)methoxy]-3,5-dimethylpyridin-2-yl}methyl)sulfinyl]-1Hbenzimidazole, sodium salt (1:1)

    2934 99 90

    376608-74-1

    2-{[(3aR,4S,6R,6aS)-6-{[5-amino-6-chloro-2-(propylsulfanyl)pyrimidin-4-yl]amino}-2,2-dimethyltetrahydro-3aH-cyclopenta[d][1,3]dioxol-4-yl]oxy}ethanol

    2934 99 90

    474554-48-8

    2-bromo-1-[3-tert-butyl-4-methoxy-5-(morpholin-4-yl)phenyl]ethanone

    2934 99 90

    530141-72-1

    3-(5-{[4-(cyclopentyloxy)-2-hydroxyphenyl]carbonyl}-2-[(3-hydroxy-1,2-benzoxazol-6-yl)methoxy]phenyl)propanoic acid

    2934 99 90

    519188-55-7

    3-[2-(1-benzothiophen-5-yl)ethoxy]-1-(3-hydroxyazetidin-1-yl)propan-1-one

    2934 99 90

    519188-42-2

    3-[2-(1-benzothiophen-5-yl)ethoxy]propionic acid

    2934 99 90

    753015-42-8

    3-{(E)-2-[(3R)-pyrrolidin-3-yl]ethenyl}-5-(tetrahydro-2H-pyran-4-yloxy)pyridine

    2934 99 90

    26638-53-9

    3-chloro-6-methyldibenzo[c,f][1,2]thiazepin-11(6H)-one 5,5-dioxide

    2934 99 90

    499785-81-8

    3-oxo-4-(2,3,5-tri-O-acetyl-β-D-ribofuranosyl)-3,4-dihydropyrazine-2-carboxamide

    2934 99 90

    356782-84-8

    3-oxo-4-(β-D-ribofuranosyl)-3,4-dihydropyrazine-2-carboxamide

    2934 99 90

    6504-57-0

    4-[3-hydroxy-3-phenyl-3-(thiophen-2-yl)propyl]-4-methylmorpholin-4-ium methyl sulfate

    2934 99 90

    871484-32-1

    4-[4-({3-[(4-deoxy-4-fluoro-b-D-glucopyranosyl)oxy]-5-(propan-2-yl)-1H-pyrazol-4-yl}methyl)phenyl]-N-[1,3-dihydroxy-2-(hydroxymethyl)propan-2-yl]butanamide

    2934 99 90

    166964-09-6

    4-chloro-3-methyl-1,2-oxazol-5-amine

    2934 99 90

    655233-39-3

    4-nitrobenzyl(6R,7R)-7-amino-8-oxo-3-[(2S)-tetrahydrofuran-2-yl]-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate hydrochloride

    2920 90 85

    89729-09-9

    5,7-dioxa-6-thiaspiro[2.5]octane-6-oxide

    2934 99 90

    388082-75-5

    5-[4-[[3-chloro-4-[(3-fluorophenyl)methoxy]phenyl]amino]-6-quinazolinyl]-2-furancarboxaldehyde – 4-methylbenzenesulfonate (1:1)

    2934 99 90

    4923-87-9

    5-bromo-1-benzothiophene

    2934 99 90

    947408-95-9

    6-(bromomethyl)-2-triphenylmethyl-1,2-benzisoxazol-3(2H)-one

    2934 99 90

    947408-94-8

    6-methyl-2-trityl-1,2-benzoxazol-3(2H)-one

    2934 99 90

    67978-05-6

    diphenylmethyl(2R)-3-methyl-2-[(1R,5S)-3-(4-methylphenyl)-7-oxo-4-oxa-2,6-diazabicyclo[3.2.0]hept-2-en-6-yl]but-3-enoate

    2934 99 90

    1001859-46-6

    DNA (synthetic plasmid vector pCOR human interferon beta signal peptide fusion protein with 21-154-human acidic fibroblast growth factor-specifying)

    2934 99 90

    665058-78-6

    DNA, d(T-sp-C-G-sp-T-sp-C-G-sp-T-sp-T-sp-T-sp-T-sp-G-sp-A-sp-C-G-sp-T-sp-T-sp-T-sp-T-sp-Gsp-T-sp-C-G-sp-T-sp-T)

    2934 99 90

    923591-06-4

    methyl (5R,7S,10S)-10-tert-butyl-15,15-dimethyl-3,9,12-trioxo-6,7,9,10,11,12,14,15,16,17,18,19-dodecahydro-1H,5H-2,23:5,8-dimethano-4,13,2,8,11-benzodioxatriazacyclohenicosine-7(3H)-carboxylate

    2934 99 90

    59337-92-7

    methyl 3-(chlorosulfonyl)thiophene-2-carboxylate

    2934 99 90

    947409-01-0

    methyl 3-[5-[4-(cyclopentyloxy)-2-hydroxybenzoyl]-2-[(2-triphenylmethyl-1,2-benzisoxazol-3(2H)-on-6-yl)methoxy]phenyl]propionate

    2934 99 90

    85006-31-1

    methyl 3-amino-4-methylthiophene-2-carboxylate

    2934 99 90

    893428-72-3

    N-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methyl-1-piperazinyl)ethoxy]-5-[(tetrahydro-2H-pyran-4-yl)oxy]-4-quinazolinamine – (2E)-2-butenedioate (1:2)

    2934 99 90

    390800-88-1

    N,N′,N′′-(boroxin-2,4,6-triyltris{[(1S)-3-methylbutane-1,1-diyl]imino[(2S)-1-oxo-3-phenylpropane-1,2-diyl]})tripyrazine-2-carboxamide

    2934 99 90

    112913-94-7

    N-{[4-(4-fluorobenzyl)morpholin-2-yl]methyl}acetamide

    2934 99 90

    120788-03-6

    S-[(1R,3S)-1-oxidotetrahydrothiophen-3-yl] ethanethioate

    2935 00 90

    1198178-65-2

    (1R,2R)-1-[(cyclopropylsulfonyl)carbamoyl]-2-ethylcyclopropanaminium 4-methylbenzenesulfonate

    2935 00 90

    39570-96-2

    (2R)-3-(benzylsulfanyl)-N-[(2S)-1-{[(2S,3S)-1-hydrazinyl-3-methyl-1-oxopentan-2-yl]amino}-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]-2-{[(4-methylphenyl)sulfonyl]amino}propanamide

    2935 00 90

    24310-36-9

    1-[(4-methylphenyl)sulfonyl]-1,2,3,4-tetrahydro-5H-1-benzazepin-5-one

    2935 00 90

    0-00-0

    2-(cyclohexylmethyl)-N-{2-[(2S)-1-methylpyrrolidin-2-yl]ethyl}-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide di[(2E)-but-2-enedioate] hydrate

    2935 00 90

    941690-55-7

    3-[(methylsulfonyl)amino]-2-phenyl-N-[(1S)-1-phenylpropyl]quinoline-4-carboxamide

    2935 00 90

    6973-09-7

    5-amino-2-methylbenzenesulfonamide

    2935 00 90

    193686-76-9

    7-chloro-1-[(4-methylphenyl)sulfonyl]-1,2,3,4-tetrahydro-5H-1-benzazepin-5-one

    2935 00 90

    123664-84-6

    N-(5-methoxy-2-phenoxyphenyl)methanesulfonamide

    2935 00 90

    149457-03-4

    N-[4-(N-formylglycyl)-5-hydroxy-2-phenoxyphenyl]methanesulfonamide

    2935 00 90

    149456-98-4

    N-[4-(N-formylglycyl)-5-methoxy-2-phenoxyphenyl]methanesulfonamide

    2935 00 90

    141450-48-8

    N-{2-[(4-hydroxyphenyl)amino]pyridin-3-yl}-4-methoxybenzenesulfonamide hydrochloride

    2935 00 90

    289042-10-0

    N-{5-[(diphenylphosphoryl)methyl]-4-(4-fluorophenyl)-6-(propan-2-yl)pyrimidin-2-yl}-N-methylmethanesulfonamide

    2939 99 00

    7689-03-4

    (4S)-4-ethyl-4-hydroxy-1H-pyrano[3′,4′:6,7]indolizino[1,2-b]quinoline-3,14(4H,12H)-dione

    2939 99 00

    477-29-2

    colchicoside

    2940 00 00

    604-69-3

    1,2,3,4,6-penta-O-acetyl-β-D-glucopyranose

    2940 00 00

    647834-15-9

    2-(4-methoxybenzyl)thiophen-3-yl β-D-glucopyranoside

    2941 90 00

    76610-92-9

    (6R,7R)-7-({N-[(4-ethyl-2,3-dioxopiperazin-1-yl)carbonyl]-D-threonyl}amino)-3-{[(1-methyl-1H-tetrazol-5-yl)sulfanyl]methyl}-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid

    3907 20 99

    913976-27-9

    poly(oxy-1,2-ethanediyl), α-hydro-ω-methoxy, diester with 21N6, 21′N6-[[(N2, N6-dicarboxy-L-lysyl-β-alanyl)imino]bis(1-oxo-2, 1-ethanediyl)]bis[N-acetylglycyl-L-leucyl-L-tyrosyl-L-alanyl-L-cysteinyl-L-histidyl-L-methionylglycyl-L-prolyl-L-isoleucyl-L-threonyl-3-(1-naphthalenyl)-L-alanyl-L-valyl-L-cysteinyl-L-glutaminyl-L-prolyl-L-leucyl-L-arginyl-N-methylglycyl-L-lysinamide] cyclic (6→15), (6′→15′) bis(disulfide)


    ANNEX IV

    List of pharmaceutical intermediates, i.e. compounds used for the manufacture of finished pharmaceutical products, to be withdrawn from the list of products receiving duty-free treatment included in Annex 6 to Annex I to Regulation (EEC) No 2658/87 due to their transfer to the list of products receiving duty-free treatment included in Annex 3 to Annex I to Regulation (EEC) No 2658/87

    CN code

    CAS RN

    Name

    2915 39 00

    2937 29 00

    7753-60-8

    17-alpha-hydroxy-3,20-dioxopregna-4,9(11)-diene-21-yl acetate

    see anecortave (INN)

    2920 90 85

    163133-43-5

    4-(nitrooxy)butyl (2S)-2-(6-methoxy-2-naphthyl) propanoate

    see naproxcinod (INN)

    2924 29 98

    194085-75-1

    2-(2-chlorophenyl)-2-hydroxyethyl carbamate

    see carisbamate (INN)

    2933 39 99

    103129-82-4

    3-ethyl 5-methyl 2-[(2-aminoethoxy)methyl]-4-(2-chlorophenyl)-6-methyl-1,4-dihydropyridine-3,5-dicarboxylate

    see levamlodipine (INN)

    2933 39 99

    319460-85-0

    N-methyl-2-{[3-((E)-2-pyridin-2-ylvinyl)-1H-indazol-6-yl]sulfanyl}benzamide

    see axitinib (INN)

    2934 10 00

    302962-49-8

    N-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)thiazole-5-carboxamide

    see dasatinib (INN)

    2934 99 90

    143491-57-0

    (2R,5S)-4-amino-5-fluoro-1-[2-(hydroxymethyl)-1,3-oxathiolan-5-yl]pyrimidin-2(1H)-one

    see emtricitabine(INN)

    2934 99 90

    98819-76-2

    (2S)-2-[(S)-(2-ethoxyphenoxy)phenylmethyl]morpholine

    see esreboxetine (INN)

    2934 99 90

    475479-34-6

    (2S)-2-methoxy-3-{4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]-1-benzothiophen-7-yl}propanoic acid

    see aleglitazar (INN)

    2934 99 90

    377727-87-2

    2-(2-furyl)-7-(2-{4-[4-(2-methoxyethoxy)phenyl] piperazin-1-yl}ethyl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[2,3-c]pyrimidin-5-amine

    see preladenant (INN)

    2934 99 90

    189003-92-7

    2-{7-fluoro-2-oxo-4-[2-(4-thieno[3,2-c]pyridin-4-ylpiperazin-1-yl)ethyl]quinolin-1(2H)-yl}acetamide

    see trelanserin (INN)

    2934 99 90

    134379-77-4

    4-amino-5-fluoro-1-[(2R,5S)-5-(hydroxymethyl)-2,5-dihydrofuran-2-yl]pyrimidin-2(1H)-one

    see dexelvucitabine (INN)

    2934 99 90

    518048-05-0

    potassium 4-[N-(2-fluorobenzyl)carbamoyl]-1-methyl-2-[1-methyl-1-(5-methyl-1,3,4-oxadiazole-2-carboxamido)ethyl]-6-oxo-1,6-dihydropyrimidine-5-olate

    see raltegravir (INN)

    2935 00 90

    170569-88-7

    4-[5-(4-fluorophenyl)-3-(trifluoromethyl)pyrazol-1-yl]benzene-1-sulfonamide

    see mavacoxib (INN)

    2935 00 90

    186497-07-4

    N-(3-methoxy-5-methylpyrazin-2-yl)-2-[4-(1,3,4-oxadiazol-2-yl)phenyl]pyridine-3-sulfonamide

    see zibotentan (INN)


    Top